许斌

创建时间:  2022/03/01  张杰   浏览次数:   返回

许斌  教授

姓名:许斌

办公室:社区学院新世纪13306

职称:教授(正高三级,博士生导师)

学历:博士

职务:社区学院副院长,九三学社上海大学委员会主委

地址:上海市宝山区上大路99号社区学院新世纪13306室,邮编:200444

电话:021-66135607

Emailxubin@t.shu.edu.cn

【教育与工作经历】

2022.2-        教授、博士生导师、社区学院副院长

2005.9-2022.1     教授、博士生导师、上海大学化学系

2002.9-2005.8     Staff Scientist,美国纽约   VivoQuest, Inc. 药物公司

2000.9-2002.8     博士后(VFA),美国国立卫生研究院(National   Institutes of Health, NIH

                            美国国立糖尿病、消化道及肾脏疾病研究所(NIDDK

                            生物有机化学及药物化学,导师:Kenneth A.   Jacobson

1997.8 2000.7     理学博士,中国科学院上海有机化学研究所

                            金属有机化学,导师:麻生明 院士

1994.8-1997.6    理学硕士,中国科学院上海有机化学研究所

                            元素有机化学,导师:朱士正 研究员

1988.9-1992.7    上海科技大学化学系

【主要获奖情况】

2020     上海市侨界杰出人物提名奖

2020     上海大学科研卓越贡献奖(理工医类)

2019      九三学社中央委员会2019年度组织工作先进个人

2019     上海市育才奖

2019     理学院科研优秀奖(2016-2019年)

2019     第十六届挑战杯全国大学生课外学术科技作品竞赛    二等奖

                《抗结直肠癌活性化合物的设计、合成与筛选》项目 指导老师

2019     九三学社上海市委社务工作先进个人

2019     上海大学年度科研创新贡献奖(年度最佳论文二等奖)

2019     第十六届挑战杯上海市大学生课外学术科技作品竞赛    一等奖

                《基于抗结直肠癌活性化合物的设计、合成与活性研究》项目 指导老师

2019     上海大学第十二届自强杯大学生课外学术科技作品竞赛 一等奖 指导老师

2018     宝钢优秀教师奖

2018     高等教育国家级教学成果二等奖(参与)

           “大国方略系列课程的创设与实践”

2018     上海大学年度科研创新贡献奖(年度最佳科研成果一等奖)

2018     上海大学年度科研创新贡献奖(年度最佳论文二等奖   3次)

2017     上海大学教学成果奖一等奖(排名第一)

2017     第十五届挑战杯全国大学生课外学术科技作品竞赛    全国特等奖

                《基于抗结直肠癌活性SGK1抑制剂的结构修饰、合成与活性研究》项目 指导老师

2017     九三学社中央委员会2013-2017年度参政议政工作先进个人

2017     上海大学年度科研创新贡献奖(年度最佳论文一等奖)

2016     Asian Core Program/Advanced Research Network Lectureship Award

2016     上海大学年度科研创新贡献奖(年度最佳论文一等奖)

2015     九三学社建社70周年上海市优秀社员

2014     Asia Core Program Lectureship Award (Singapore)

2011     上海大学理学院研究生导师优秀奖   (2009 - 2011学年)

2009     上海大学理学院研究生导师优秀奖   (2007 - 2009学年)

2009     上海大学毕业生初次就业率贡献奖

2009     上海大学十佳杰出青年提名奖

2007     上海市浦江人才计划

2002     上海市科技进步二等奖

2000     美国NIH   Visiting Fellow Award

2000     中国科学院刘永龄奖学金博士一等奖

【主持的主要科研项目】

1.    异腈参与的惰性化学键可控转化

国家自然科学基金委员会(2022.0160   2025.12

2.    基于廉价硝酸铜的可控化学转化与含氮杂环构建

国家自然科学基金 (No. 21871174) (2019.12022.12)

3.    基于廉价铜盐阴离子的精准合成及其在心肌纤维化防治中的应用

上海市教育委员会科研创新计划非共识项目   (2019-01-07-00-09-E00008) (2019.12023.12)

4.    异腈参与的惰性键活化与含氮杂环构建

国家自然科学基金 (No. 21672136) (2017.12020.12)

5.    基于氧化胺化反应的含氮杂环合成

国家自然科学基金 (No. 21272149) (2013.12016.12)

6.    基于惰性化学键活化的含氮杂环合成

上海市教委科研创新重点项目 (No.14ZZ094) (2014.012016.12)

7.    金属催化的1,1-二溴-1-烯烃的多中心反应研究

国家自然科学基金 (No. 20972093) (2010.12012.12)

8.    含氮杂环中的多碳-氮键形成反应研究

国家自然科学基金 (No. 20672071) (2007.12009.12)

9.    抗丙肝病毒含氮分子库的定向多样性合成及活性研究

上海市浦江人才计划 (No. 07pj14043)   (2007.102009.9)

【主要研究领域】

1. 惰性化学键可控转化

2. 新型药物分子设计及合成

【近期主要论文著作】

68. Cun Yang, Zhi-Xiong Yang,   Chang-Hua Ding,* Bin Xu, and Xue-Long Hou*

Development of Dipolarophiles for   Catalytic Asymmetric Cycloadditions through Pd-π-allyl zwitterions

Chem. Rec. 2021,   ASAP [Link].

67. Weixiang Wang, Tianqi Liu, Chang-Hua   Ding,* and Bin Xu*

C(sp3)–H Functionalization with Isocyanides

Org. Chem. Front.,   2021, ASAP. [Link]

66. Jimin Guo, Jianjian Zha, Tao   Zhang, Chang-Hua Ding, Qitao Tan,* Bin Xu*

PdCl2/DMSO-Catalyzed   Thiol–Disulfide Exchange: Synthesis of Unsymmetrical Disulfide

Org. Lett,   2021, 23, 3167–3172 [Link]

65.α-Iminonitriles: Composite   Functional Groups for Functionalization of Pyrene

Guigang Deng, Tianqi Liu, Yuqin   Wang, Bingxin Liu, Qitao Tan,* Bin Xu,*

Asian J. Org. Chem.   2021, 10, 262-272. [Linker].

64. Tianyin Huang, Yang Yu, Hui   Wang, Yifan Lin, Yurui Ma, Haoyu Wang, Chang-Hua Ding,* Junjie Xiao,* Bin   Xu,*

Silver-Promoted Regioselective   Oxidative Decarboxylative C–H Alkylation of Phenanthridines with Carboxylic   Acids

Synthesis   2020, 52, 239–245. [Linker].

63. Juan Du, Yuan-Da Hua, Yang-Jie   Jiang, Shuai Huang, Di Chen, Chang-Hua Ding,* Xue-Long Hou,*

Palladium-Catalyzed Asymmetric   Decarboxylative [4+2] Dipolar Cycloaddition of 4 Vinyl-1,3-dioxan-2-ones with   α,β-Disubstituted Nitroalkenes Enabled by a Benzylic Substituted P,N-Ligand

Org. Lett.   2020, 22, 53755379.   [Linker].

62. Leiyang Zhao, Bingxin Liu,   Qitao Tan, Chang-Hua Ding*, Bin Xu*

"Silver-Assisted Oxidative   Isocyanide Insertion of Ethers: A Direct Approach to β-Carbonyl   α-Iminonitriles"

Org. Lett.   2019, 21, 9223-9227.

61. Huiwen Chi, Hao Li, Bingxin Liu,   Rongxuan Ye, Haoyang Wang, Yin-Long Guo, Qitao Tan* and Bin Xu*

“From Isocyanides to Iminonitriles   via Silver-Catalyzed Sequential Insertion of C(sp3)–H Bond”

iScience,   2019, 21, 650-663.

60. Tianyi Huang, Yang Yu, Hui   Wang, Yifan Lin, Yurui Ma, Haoyu Wang, Chang-Hua Ding,* Junjie Xiao,* Bin Xu,*

“Silver-Promoted Oxidative   Decarboxylative C–H Alkylation of Phenanthridines with Carboxylic Acids”

Synthesis   2019, 51, DOI: 10.1055/s-0039-1690220.

59. Mengjing Jiang, Jimin Guo,   Bingxin Liu, Qitao Tan,* and Bin Xu,*

“Synthesis of Tellurium-Containing   π-Extended Aromatics with Room-Temperature Phosphorescence”

Org. Lett.   2019, 21, 8328-8333.

58. Mingchun Gao, Yuansheng Gan,   and Bin Xu*

"From Alkenes to Isoxazolines   via Copper-Mediated Alkene Cleavage and Dipolar Cycloaddition"

Org. Lett.,   2019, 21, 7435-7439.

57. Haoyu Wang, Yurui Ma, Yifan   Lin, Jiajie Liu, Rui Chen, Bin Xu,* Yajun Liang,,*

"An Isoxazole Derivative   SHU00238 Suppresses Colorectal Cancer Growth through miRNAs Regulation"

Molecules   2019, 24, 2335. (Special Issue Anti-Cancer Drug: Discovery,   Development and Combination)

56. Ze-Zhen Jiang, Yang-Jie Jiang,   Juan Du, Di Chen, Chang-Hua Ding*, Bin Xu*, Xue-Long Hou*

"Palladium-Catalyzed Asymmetric   Heck-Matsuda Reaction of 1,4-Dihydroquinolines with Aryldiazonium Salts"

Synthesis   2019, 51, 3269-3276.

55. Yifan Lin, Ke Zhang, Mingchun   Gao, Zheyi Jiang, Jiajie Liu, Yurui Ma, Haoyu Wang, Qitao Tan*, Junjie Xiao*   and Bin Xu*

"Copper nitrate-mediated   synthesis of 3-aryl isoxazolines and isoxazoles from olefinic   azlactones"

Org. Biomol. Chem.,   2019, 17, 5509–5513.

54. Mingchun Gao, Kaijing Zhou, and   Bin Xu

"Copper Nitrate-Mediated   Selective Difunctionalization of Alkenes: A Rapid Access to   β-Bromonitrates"

Adv. Synth. Catal.   2019, 361, 2031-2036.

53. Mingchun Gao, Minfen Zou, Jue   Wang, Qitao Tan, Bingxin Liu, and Bin Xu*

"Palladium-Catalyzed   Multicomponent Reaction of Alkynes, Carboxylic Acids, and Isocyanides: A   Direct Approach to Captodative Olefins"

Org. Lett.,   2019, 21, 1596-1597.

52. Tao Zhang, Guigang Deng, Hanjie   Li, Bingxin Liu, Qitao Tan,* and Bin Xu*

"Cyclization of   2-biphenylthiols to dibenzothiophenes under PdCl2/DMSO catalysis"

Org. Lett.,   2018, 20, 5439-5443.

51. Jian-Guo Liu, Wen-Wen Chen,*   Chang-Xue Gu, Bin Xu,* Ming-Hua Xu*

"Access to Spiroindolines and   Spirodihydrobenzofurans via Pd-Catalyzed Domino Heck Spiroyclization through   C-H Activation and Carbene Insertion"

Org. Lett.,   2018, 20, 2728-2732.

50. Zhuang Tian, Jiaojiao Xu,   Bingxin Liu, Qitao Tan,* Bin Xu,*

"Copper-Catalyzed Synthesis of   Polysubstituted Pyrroles through [3+1+1] Cycloaddition Reaction of Nitrones   and Isocyanides"

Org. Lett.,   2018, 20, 2603-2606.

49. Mingchun Gao, Rongxuan Ye,   Weijia Shen and Bin Xu*

"Copper nitrate: a privileged   reagent for organic synthesis"

Org. Biomol. Chem.,   2018, 16, 2602-2618. (Invited Review)

48. Chunling Lan, Zhuang Tian,   Xuchun Liang, Mingchun Gao, Wenting Liu, Yu An, Wencheng Fu, Guanming Jiao,   Junjie Xiao, and Bin Xu*  

"Copper-Catalyzed Aerobic   Annulation of Hydrazones: Direct Access to Cinnolines"

Adv. Synth. Catal.,   2017, 359, 3735-3740.

47. Ze-Zhen Jiang, Ang Gao, Hao Li,   Di Chen, Chang-Hua Ding*, Bin Xu*, Xue-Long Hou*

"Enantioselective Synthesis of   Chromenes via a Palladium-Catalyzed Asymmetric Redox-Relay Heck   Reaction"

Chem. Asian J.,   2017, 12, 3119-3122.

46. Tengda Si, Bowen Li, Wenrui   Xiong, Bin Xu,* and Wenjun Tang,*

"Efficient cross-coupling of   aryl/alkenyl triflates with acyclic secondary alkylboronic acids"

Org. Biomol. Chem.,   2017, 15, 9903-9909.

45. Qitao Tan*, Dandan Zhou, Tao   Zhang, Bingxin Liu, Bin Xu*

"Iodine-doped Sumanene and Its   Application for the Synthesis of Chalcogenasumanenes and    Silasumanenes"

Chem Commun.   2017, 53, 10279-10282.

44. Dandan Zhou, Ya Gao, Bingxin   Liu, Qitao Tan*, Bin Xu,*

"Synthesis of Silicon and   Germanium-Containing Heterosumanenes via Rhodium-Catalyzed Cyclodehydrogenation   of Silicon/Germanium–Hydrogen and Carbon–Hydrogen Bonds"

Org. Lett.   2017, 19, 4628-4631.

43. Zong-Feng Zhang, Dong-Xing Zhu,   Wen-Wen Chen, Bin Xu*, Ming-Hua Xu*

"Enantioselective Synthesis of   gem-Diaryl Benzofuran-3(2H)-ones via One-Pot Asymmetric Rhodium/Palladium   Relay Catalysis"

Org. Lett.   2017, 19, 2726-2729.

42. Xiaohu Hong, Qitao Tan, Bingxin   Liu, Bin Xu*

"Isocyanide Induced Activation   of Copper Sulfate: Direct Access to Functionalized Heteroarene Sulfonic   Esters"

Angew. Chem., Int. Ed.   2017, 56, 3961-3965.

41. Yingying Li, Mingchun Gao,   Bingxin Liu, Bin Xu*

"Copper Nitrate-Mediated   Chemo- and Regioselective Annulation from Two Different Alkynes: A Direct   Route to Isoxazoles"

Org. Chem. Front.   2017, 4, 445-449.

40. Bingrui Song, Bin Xu*

"Metal-catalyzed C–H   functionalization involving isocyanides"

Chem. Soc. Rev.,   2017, 46, 1103-1123. (封面论文)

39. Hao Li, Ang Gao, Xiu-Yan Liu,   Chang-Hua Ding*, Bin Xu*, Xue-Long Hou*

"Kinetic Resolution of   5-Substituted-Cyclohexenols by Pd-Catalyzed Asymmetric Redox-Relay Heck   Reaction"

Synthesis   2017, 49, 159-166.

38. Mingchun Gao, Bin Xu*

"Copper Nitrate-Mediated   Regio- and Stereoselective Difunctionalization of Alkynes: A Direct Approach   to a-Chloro-β-nitroolefins"

Org. Lett.   2016, 18, 4746-4749.

37. Xu Zhang, Bin Xu* and Ming-Hua   Xu*

"Rhodium-catalyzed asymmetric   arylation of N- and O-containing cyclic aldimines: facile and efficient   access to highly optically active 3,4-dihydrobenzo[1,4]oxazin-2-ones and   dihydroquinoxalinones"

Org. Chem. Front.,   2016, 3, 944-948.

36. Qitao Tan and Bin Xu,*

"CH   Bond Activation as a Powerful Tool in the Construction of Biologically Active   Nitrogen Containing Heterocycles"

Studies in Natural   Products Chemistry, 2016, 50,   299-340. (Invited book chapter).

35. Mingchun Gao and Bin Xu,*

"Transition Metal-Participated   Synthesis and Utilization of N-containing Heterocycles: Exploring for Nitrogen   Sources"

Chem. Rec.   2016, 16, 1701-1714. (个人研究综述)

34. Hong Mao, Mingchun Gao, Bingxin   Liu and Bin Xu,*

"Manganese(II)-catalyzed   modular synthesis of isoquinolines from vinyl isocyanides and   hydrazines"

Org. Chem. Front.   2016, 3, 516-521.

33. Qitao Tan,* Huanhuan Chen,   Huaida Xia, Bingxin Liu and Bin Xu,*

"Parent and Trisubstituted   Triazacoronenes: Synthesis, Crystal Structure and Physicochemical   Properties"

Chem. Commun.   2016, 52, 537-540.

国内外媒体亮点推介:SynfactsX-Mol.

32. Hao Li, Shi-Li Wan, Changhua Ding,*   Bin Xu* and Xue-Long Hou

"Kinetic Resolution of   2-Substituted-2,3-dihydrofurans by Palladium-Catalyzed Asymmetric Heck "

RSC Advances   2015, 5, 75411-75414.

31. Mingchun Gao, Yingying Li,   Yuansheng Gan and Bin Xu*

"Copper Nitrate-Mediated   Regioselective [2+2+1] Cyclization of Alkynes with Alkenes: A Cascade   Approach to Δ2-Isoxazolines"

Angew. Chem., Int. Ed.,   2015, 54, 8795-8799. (封面论文)

国内外媒体亮点推介:Synfacts;中国科学报;教育部科技发展中心;科学网;X-Mol

30. Zhengwei Ding, Qitao Tan*, Bingxin   Liu, Ke Zhang, Bin Xu*

"Copper-Promoted Oxidative CH   Bond Amination of Hydrazones: Synthesis of 1H-Indazoles and   1H-Pyrazoles"

Acta Chimica Sinica,   2015, 73, 1302-1306. (主编邀请稿,   Special topic: C-H activation)    

29. Diao Chen, Xu Zhang, Wei-Yi Qi,   Bin Xu and Ming-Hua Xu*

"Rhodium(I)-Catalyzed   Asymmetric Carbene Insertion into BH   Bonds: Highly Enantioselective Access to Functionalized Organoboranes"

J. Am. Chem. Soc.,   2015, 137, 5268–5271. (封面论文)

28. Zhengwei Ding, Qitao Tan,   Mingchun Gao and Bin Xu*

"Copper-catalyzed Aerobic   Cascade Cycloamination and Acyloxylation: a Direct Approach to   4-Acyloxy-1H-pyrazoles"

Org. Biomol. Chem.   2015, 13, 4642-4646.

27. Hao Wang and Bin Xu*

"Recent Advances in Inert   Bonds Activation with Isocyanides"

Chin. J. Org. Chem.   2015, 35, 588-602. (主编邀请综述)

26. Hao Li, Changhua Ding*, Bin   Xu*, Xuelong Hou*

"Recent Developments in   Palladium-Catalyzed Asymmetric Intermolecular Heck Reaction"

Acta Chimica Sinica,   2014, 72, 765-770. (Review)  

25. Guangyin Qian, Xiaohu Hong,   Bingxin Liu, Hong Mao and Bin Xu*

"Rhodium-catalyzed   Regioselective C–H Chlorination of 7- Azaindoles Using   1,2-Dichloroethane"

Org. Lett.   2014, 16, 5294-5297.

24. Xiaohu Hong, Hao Wang, Bingxin   Liu and Bin Xu*

"Ruthenium-Catalyzed   Double-Fold C-H Tertiary Alkoxycarbonylaton Arenes Using Di-tert-butyl   Dicarbonate"

Chem Commun.   2014, 50, 14129-14132.

23. Hao Wang, Yang Yu, Xiaohu Hong   and Bin Xu*

"Mn(II)/O2-Promoted Oxidative   Annulation of Vinyl Isocyanides with Boronic Acids: Synthesis of Multi-substituted   Isoquinolines"

Chem Commun.   2014, 50, 13485-13488.

22. Guangyin Qian, Bingxin Liu,   Qitao Tan, Siwen Zhang, and Bin Xu*

"Hypervalent   Iodine(III)-Promoted Direct Synthesis of Imidazo[1,2-a]pyrimidines"

Eur. J. Org. Chem.   2014, 2014, 4837-4843.

21. Tao Fang, Qitao Tan, Zhengwei   Ding, Bingxin Liu and Bin Xu*

" Pd-Catalyzed Oxidative Annulation   of Hydrazides with Isocyanides: Synthesis of 2-Amino-1,3,4-oxadiazoles"

Org. Lett.   2014, 16, 2342-2345. Highlighted by   Org. Chem. Portal 网站

20. Hao Wang, Yang Yu, Xiaohu Hong,   Qitao Tan and Bin Xu*

" Rhodium-Catalyzed Direct   ortho C–N Bond Formation of Aromatic Azo Compounds with Azides"

J. Org. Chem.   2014, 79, 3279-3288.

19. Xiaohu Hong, Hao Wang, Guangyin   Qian, Qitao Tan and Bin Xu*

" Rhodium-Catalyzed Direct C–H   Bond Cyanation of Arenes with Isocyanide"

J. Org. Chem.   2014, 79, 3228-3237.

18. Xiaomei Huang, Shuguang Xu,   Qitao Tan, Mingchun Gao, Minjie Li and Bin Xu*

"Copper-mediated Tandem   Reaction through Isocyanides N–H Bond Insertion: Efficient Access to   Unsymmetrical Tetrasubstituted Ureas"

Chem Commun.   2014, 50, 1465-1468.

17. Jie Sun, Qitao Tan, Wusong   Yang, Bingxin Liu and Bin Xu*

“Copper-Catalyzed Aerobic Oxidative   Annulation and Carbon-Carbon Bond Cleavage of Arylacetamides: Domino   Synthesis of Fused Quinazolinones”

Adv. Synth. Catal.   2014, 356, 388-394.

16. Wenting Liu, Xiaohu Hong, Bin   Xu*

"Rhodium-Catalyzed Oxidative   Coupling of Aryl Hydrazones with Internal Alkynes: Efficient Synthesis of   Multisubstituted Isoquinolines" (主编邀请稿,   Special topic: Rhodium catalysis)

Synthesis 2013,   45, 2137-2149.

15. Jie Sun, Bingxin Liu, and Bin   Xu*

"Copper-Catalyzed Tandem   Oxidative Cyclization of Arylacetamides: Efficient Access to N- Functionalized   Isatins"

RSC Advances   2013, 3, 5824-5827.

14. Guifei Li, Zhengwei Ding, and   Bin Xu*

"Rhodium-Catalyzed Oxidative   Annulation of Sulfonylhydrazones with Alkenes"

Org. Lett.   2012, 14, 5338-5341.  

13. Shuguang Xu, Xiaomei Huang,   Xiaohu Hong, and Bin Xu*

"Palladium-Assisted   Regioselective C–H Cyanation of Heteroarenes Using Isonitrile as Cyanide   Source"

Org. Lett.   2012, 14, 4614-4617.  

12. Bingxin Liu, Xiaohu Hong, Dong   Yan, Shuguang Xu, Xiaomei Huang, and Bin Xu*

"Palladium-Catalyzed Tandem   Allenyl and Aryl C–N Bond Formation: Efficient Access to N-Functionalized   Multi-substituted Indoles"

Org. Lett.   2012, 14, 4398-4401.  

11. Jun Shao, Xiaomei Huang, Xiaohu   Hong, Bingxin Liu and Bin Xu*

"Synthesis of N–Alkyl   Substituted 4-Quinolones via Tandem Alkenyl and Aryl C–N Bond   Formation"  (主编邀请稿, Special topic: Tandem   reaction)

Synthesis   2012, 44, 1798-1808. Highlighted by Org. Chem. Portal 网站

10. Jun Shao, Xiaomei Huang, Siyuan   Wang, Bingxin Liu, Bin Xu*

"A straightforward synthesis   of N-monosubstituted a-keto amides via aerobic benzylic oxidation of   amides"

Tetrahedron   2012, 68, 573-579.

9. Chengming Wang, Caiyun Sun, Fei   Weng, Mingchun Gao, Bingxin Liu and Bin Xu*

"Unexpected formation of   (Z)-3-(halomethylene) isoindolinones from gem-dihalovinylbenzonitriles:   Efficient synthesis of enyne-containing isoindolinones"

Tetrahedron Lett.   2011, 52, 2984-2989.      

8. Xiaojian Zheng, Bingrui Song,   Guifei Li, Bingxin Liu, Hongmei Deng and Bin Xu*

"Direct synthesis of   ortho-dihalogenated arylpyrimidines using calcium halides as halogen   sources"

Tetrahedron Lett.   2010, 51, 6641-6645.    

7. Xiaojian Zheng, Bingrui Song and   Bin Xu*

"Palladium-Catalyzed   Regioselective C-H Bond ortho-Acetoxylation of Arylpyrimidines"

Eur. J. Org. Chem.   2010, 4376-4380.      

6. Fei Weng, Chengming Wang and Bin   Xu*

"Direct C-H bond arylation of   2-hydroxybenzaldehydes with arylboronic acids via ligand-free palladium   catalysis"

Tetrahedron Lett.   2010, 51, 2593-2596.    

5. Bingrui Song, Xiaojian Zheng,   Jun Mo and Bin Xu*

"Palladium-Catalyzed   Monoselective Halogenation of C-H Bonds: Efficient Access to halogenated   Arylpyrimidines using Calcium Halides"

Adv. Synth. Catal.   2010, 352, 329-335.    

4. Tiankun Zhao and Bin Xu*

"Palladium-Catalyzed Tandem   Amination Reaction for the Synthesis of 4-Quinolones"

Org. Lett.   2010, 12, 212-215.    

Highlighted by Synfacts 2010, 4,   0408.

Highlighted by Org. Chem. Portal 网站

3. Wenchao Ye, Jun Mo, Tiankun Zhao   and Bin Xu*

"Palladium-Catalyzed   Amidation-Hydrolysis Reaction of gem-Dihaloolefins: Efficient Synthesis of   Homologated Carboxamides from Ketones"

Chem Commun.   2009, 3246-3248.    

Highlighted by Org. Chem. Portal 网站;   see, D. F. Taber, Org. Chem. Highlights 2010, March 22.

2. Caiyun Sun and Bin Xu*

"A Tandem   Elimination-Cyclization-Suzuki Approach: Efficient One-pot Synthesis of   Functionalized (Z)-3-(Arylmethylene)isoindolin-1-ones"

J. Org. Chem.   2008, 73, 7361-7364.  

1. Bingrui Song, Siyuan Wang,   Caiyun Sun, Hongmei Deng and Bin Xu*

"Cesium Carbonate Promoted   Aerobic Oxidation of Arylacetamides: An Efficient Access to N-Substituted   a-keto amides"

Tetrahedron Lett.   2007, 48, 8982-8986.

【授权国外专利】

1. Bin Xu, Qiang Zhu, Hyun-Joon   Cho; Reza Fathi, Zhen Yang, Anthony Sandrasagra, Yixin Liu, "3,   4-Disubstituted coumarin and quinolone compounds for the treatment of   hepatitis C virus infection" Pub. No.: US 2006/0223783 A1 (Pub. Date:   Oct. 5, 2006); WO 2007133211 A1 (Pub. Date: Nov. 22, 2007)

2. Youhong Hu, Bin Xu, Yun Liao,   Kenneth Nawoschik, Yixin Liu, Anthony Sandrasagra, Reza Fathi, Zhen Yang,   "Preparation of pyrazole derivatives for treatment of hepatitis C virus   infection" Pub. No.: US 2006/0183751 A1 (Pub. Date: Aug. 17, 2006); WO 2006088903   A2 (Pub. Date: Aug. 24, 2006)

【学生培养】

蔺一凡    第十六届挑战杯上海市大学生课外学术科技作品竞赛    一等奖 2019年)

蔺一凡    上海大学第十二届自强杯大学生课外学术科技作品竞赛 一等奖 2019年)

兰春岭    上海大学校长奖 2019年)

兰春岭    宝钢优秀学生奖 2018年)

兰春岭    第十五届挑战杯全国大学生课外学术科技作品竞赛    全国特等奖(2017年)

       第十五届挑战杯全国大学生课外学术科技作品竞赛    全国特等奖(2017年)

周丹丹    国家奖学金(硕士) 2017年)

周丹丹    上海大学研究生创新奖 2017年)

周丹丹    国家学业奖学金硕士一等奖 2017年)

洪小虎    19届全国金属有机化学学术讨论会最佳墙报奖 2016年)

高明春    国家奖学金(博士) 2016年)

高明春    上海大学光华奖学金博士一等奖(2015年)

高明春    国家学业奖学金博士一等奖 2015年)

陈欢欢    国家学业奖学金硕士一等奖 2015年)

洪小虎    国家奖学金(博士) 2014年)

洪小虎    上海大学光华奖学金博士一等奖 2014年)

       国家奖学金(硕士) 2014年)

       上海大学光华奖学金硕士一等奖 2014年)

       国家学业奖学金硕士一等奖 2014年)

钱光印    18届全国金属有机化学学术讨论会最佳墙报奖 2014年)

刘文婷    上海市优秀毕业生    2014年)

       上海大学今井嘉夫奖学金 2014年)

钱光印    上海大学陈念贻奖学金    2014年)

刘文婷    上海大学光华奖学金硕士二等奖     2013年)

刘文婷    上海大学优秀学生 2012年)

孙彩云    上海市研究生优秀成果(学位论文) 2011年)

宋炳瑞    上海市研究生优秀成果(学位论文) 2011年)

李贵飞    上海大学研究生创新基金    2011年)

刘文婷    上海大学感动上大人物”   20092010年度)

郑晓建    上海大学光华奖学金硕士二等奖 2010年)

       上海大学第九届英语演讲比赛暨

                "外研社杯"全国英语演讲选拔赛优胜奖    2010年)

赵添堃    上海大学今井嘉夫奖学金    2010年)

郑晓建    上海大学研究生创新基金 2010年)

孙彩云    上海大学优秀毕业生     2009年)

       上海大学研究生创新基金    2009年)

孙彩云    上海大学光华奖学金硕士一等奖    2008年)

宋炳瑞    上海大学光华奖学金硕士二等奖    2008年)

【社会服务与兼职】

九三学社上海大学委员会  主委

上海市宝山区政协委员

九三学社上海市委员会  教育专门委员会委员

上海市欧美同学会上海大学分会  副会长

上海市第六批党外挂职干部(宝山基地)

 

中国中药协会微循环用药专业委员会   常务委员

中国中药协会心血管药物研究专业委员会   委员

 

以色列国家基金委、国家基金委、国家留学基金委、上海市科委项目评审专家

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